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Found 2 Enz. Inhib. hit(s) with Target = 'Arachidonate 5-lipoxygenase-activating protein' and Ligand = 'BDBM50383917'
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50383917(CHEMBL2031658)
Affinity DataIC50:  1.10nMAssay Description:Displacement of [125I]L-691,831 from 5-lipoxygenase-activating protein in human polymorphonuclear cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetArachidonate 5-lipoxygenase-activating protein(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50383917(CHEMBL2031658)
Affinity DataIC50:  375nMAssay Description:Inhibition of 5-lipoxygenase-activating protein in human polymorphonuclear cells assessed as inhibition of calcium ionophore-induced LTB4 production ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed