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Found 3 Enz. Inhib. hit(s) with Target = 'Aromatase' and Ligand = 'BDBM8916'
TargetAromatase(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM8916(1-(2-Naphthyl)-1H-imidazole | 1-(naphthalen-2-yl)-...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of aromataseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM8916(1-(2-Naphthyl)-1H-imidazole | 1-(naphthalen-2-yl)-...)
Affinity DataIC50:  2.82E+3nMAssay Description:The enzyme activity was assayed by measuring the 3H-labeled H2O formed from [1beta-3H] Androstenedione during aromatization. After incubation, the re...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM8916(1-(2-Naphthyl)-1H-imidazole | 1-(naphthalen-2-yl)-...)
Affinity DataIC50:  2.82E+3nMpH: 7.4Assay Description:The enzyme was obtained from the microsome fraction of fresh human placenta (St. Josephs Krankenhaus, Saarbrucken-Dudweiler, Germany) according to th...More data for this Ligand-Target Pair
In DepthDetails US Patent