Affinity DataKi: 0.400nMAssay Description:Displacement of [3H]des-arg10, leu9-kallidin from human bradykinin B1 receptor expresed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.690nMAssay Description:Binding affinity to rabbit bradykinin B1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 35.3nMAssay Description:Displacement of [3H]des-arg10 kallidin from rat bradykinin B1 receptor expresed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.25nMAssay Description:Antagonist activity at bradykinin B1 receptor expresed in CHO cells assessed as inhibition of des-arg10-kallidin-induced increase in cytosolic calciu...More data for this Ligand-Target Pair
Affinity DataIC50: 2.40nMAssay Description:Activity at rabbit bradykinin B1 receptor assessed by FLIPR assayMore data for this Ligand-Target Pair