Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) with Target = 'B1 bradykinin receptor' and Ligand = 'BDBM50309020'
TargetB1 bradykinin receptor(Homo sapiens (Human))
Jerini

Curated by ChEMBL
LigandPNGBDBM50309020(CHEMBL605634 | methyl 4'-((1H-benzo[d]imidazol-2-y...)
Affinity DataIC50:  3.50E+3nMAssay Description:Antagonist activity at bradykinin B1 receptor in human IMR90 cells pretreated with IL1beta assessed as inhibition of DAKD-induced calcium mobilizatio...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed