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Found 3 Enz. Inhib. hit(s) with Target = 'B2 bradykinin receptor' and Ligand = 'BDBM50435301'
TargetB2 bradykinin receptor(Homo sapiens (Human))
Institute Of Organic Synthesis

Curated by ChEMBL
LigandPNGBDBM50435301(CHEMBL446325 | NPC-567)
Affinity DataIC50:  10nMAssay Description:Binding affinity to human bradykinin B2 receptor by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Institute Of Organic Synthesis

Curated by ChEMBL
LigandPNGBDBM50435301(CHEMBL446325 | NPC-567)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]bradykinin from human recombinant bradykinin B2 receptor expressed in CHO cells measured after 60 mins by scintillation counting ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetB2 bradykinin receptor(Homo sapiens (Human))
Institute Of Organic Synthesis

Curated by ChEMBL
LigandPNGBDBM50435301(CHEMBL446325 | NPC-567)
Affinity DataIC50:  14nMAssay Description:Displacement of [3H]bradykinin from human recombinant B2 bradykinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed