Found 3 Enz. Inhib. hit(s) with Target = 'BTB/POZ domain-containing protein KCTD12' and Ligand = 'BDBM50505532'
TargetBTB/POZ domain-containing protein KCTD12(Homo sapiens)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataKi: 840nMAssay Description:Displacement of TAMRA-AAG-SLQLPILHHAYLPSIGGV from recombinant human 6X His-tagged KCTD12 T1 domain (27 to 131 residues) expressed in Escherichia coli...More data for this Ligand-Target Pair
TargetBTB/POZ domain-containing protein KCTD12(Homo sapiens)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataIC50: 4.82E+3nMAssay Description:Displacement of TAMRA-AAG-SLQLPILHHAYLPSIGGV from recombinant human 6X His-tagged KCTD12 T1 domain (27 to 131 residues) expressed in Escherichia coli...More data for this Ligand-Target Pair
TargetBTB/POZ domain-containing protein KCTD12(Homo sapiens)
University Of Copenhagen
Curated by ChEMBL
University Of Copenhagen
Curated by ChEMBL
Affinity DataEC50: 300nMAssay Description:Binding affinity to recombinant human 6X His-tagged KCTD12 T1 domain (27 to 131 residues) expressed in Escherichia coli BL21 DE3 cells preincubated f...More data for this Ligand-Target Pair