TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKi: 1.00E+3nMAssay Description:Displacement of [3H]CGP12177 from human beta2 adrenoceptor expressed in CHO cell membranesMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataEC50: 1.00E+4nMAssay Description:Agonist activity at human beta2 adrenoceptor expressed in CHOK1 cells assessed as induction of [3H]cAMP accumulation after 5 hrsMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKd: 1.45E+3nMAssay Description:Displacement of [3H](-)CGP12177 from human beta2-AR expressed in CHOK1 cells after 2 hrs by TopCount microscintillation counting methodMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKd: 1.05E+3nMAssay Description:Antagonist activity at human beta2 adrenoceptor expressed in CHOK1 cells assessed as inhibition of cimaterol-induced [3H]cAMP accumulation incubated ...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKd: 776nMAssay Description:The whole cell-binding studies were undertaken in CHO cell lines stably expressing each beta-adrenoceptor subtype. Nonspecific binding was determined...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Friedrich-Alexander Universit£T Erlangen-N£Rnberg
Curated by ChEMBL
Affinity DataKd: 1.51E+3nMAssay Description:Displacement of [3H]-CGP12177 from human beta2 adrenoceptor expressed in CHOK1 cells after 2 hrs by scintillation counting analysisMore data for this Ligand-Target Pair