TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Institute Of Cell Signaling
Curated by PDSP Ki Database
Institute Of Cell Signaling
Curated by PDSP Ki Database
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Institute Of Cell Signaling
Curated by PDSP Ki Database
Institute Of Cell Signaling
Curated by PDSP Ki Database
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Institute Of Cell Signaling
Curated by PDSP Ki Database
Institute Of Cell Signaling
Curated by PDSP Ki Database
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Institute Of Cell Signaling
Curated by PDSP Ki Database
Institute Of Cell Signaling
Curated by PDSP Ki Database
Affinity DataEC50: 3.16E+3nMAssay Description:Agonist activity at human adrenergic beta2 receptor expressed in H292 cells assessed as intracellular cAMP accumulation after 1 hrMore data for this Ligand-Target Pair
Affinity DataKd: 3.98E+3nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
Affinity DataKd: 1.86E+3nMAssay Description:Affinity for cow beta-2 adrenergic receptor by measuring displacement (-)-[3H]dihydroalprenolol (DHA)More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Institute Of Cell Signaling
Curated by PDSP Ki Database
Institute Of Cell Signaling
Curated by PDSP Ki Database
Affinity DataKd: 2.51E+3nMAssay Description:Binding affinity to beta-2 adrenergic receptor (unknown origin) at 1 to 10000 nMMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Institute Of Cell Signaling
Curated by PDSP Ki Database
Institute Of Cell Signaling
Curated by PDSP Ki Database
Affinity DataKd: 3.20nMAssay Description:Displacement of [3H]-CGP12,177 from immobilized Halo tag-fused beta2 adrenoceptor (unknown origin) expressed in Escherichia coli BL21 (DE3)More data for this Ligand-Target Pair
Affinity DataKd: 4.48E+3nMAssay Description:Apparent binding affinity constant to beta-2 adrenergic receptor determined using [3H]DHAMore data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Institute Of Cell Signaling
Curated by PDSP Ki Database
Institute Of Cell Signaling
Curated by PDSP Ki Database
Affinity DataKd: 2.40E+3nMAssay Description:The whole cell-binding studies were undertaken in CHO cell lines stably expressing each beta-adrenoceptor subtype. Nonspecific binding was determined...More data for this Ligand-Target Pair
TargetBeta-2 adrenergic receptor(Homo sapiens (Human))
Institute Of Cell Signaling
Curated by PDSP Ki Database
Institute Of Cell Signaling
Curated by PDSP Ki Database
Affinity DataKd: 2.51E+3nMAssay Description:Binding affinity to human adrenergic beta2 receptorMore data for this Ligand-Target Pair