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Found 2 Enz. Inhib. hit(s) with Target = 'Beta-3 adrenergic receptor' and Ligand = 'BDBM50076960'
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50076960(4-[4-(3-Cyclopentyl-propyl)-5-oxo-4,5-dihydro-tetr...)
Affinity DataIC50:  92nMAssay Description:Inhibitory activity against cloned human Beta-3 adrenergic receptor in the presence of [125I]-iodocyanopindolol expressed in CHO cells by receptor bi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50076960(4-[4-(3-Cyclopentyl-propyl)-5-oxo-4,5-dihydro-tetr...)
Affinity DataEC50:  13nMAssay Description:Agonistic activity against the cloned human Beta-1 adrenergic receptor was measured by its by its ability to stimulate adenylyl cyclaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed