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Found 5 Enz. Inhib. hit(s) with Target = 'Beta-lactamase' and Ligand = 'BDBM50212641'
TargetBeta-lactamase(Proteus mirabilis)TBA
LigandPNGBDBM50212641(Brobactam)
Affinity DataIC50:  3.57nMAssay Description:Inhibitory activity against Proteus vulgaris HJ33C Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
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TargetBeta-lactamase(Staphylococcus aureus)TBA
LigandPNGBDBM50212641(Brobactam)
Affinity DataIC50:  46.4nMAssay Description:Inhibitory activity against Staphylococcus aureus CJ8 beta-lactamase enzymeMore data for this Ligand-Target Pair
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TargetBeta-lactamase(Klebsiella oxytoca)TBA
LigandPNGBDBM50212641(Brobactam)
Affinity DataIC50:  285nMAssay Description:Inhibitory activity against Klebsiella oxytoca HC7 Class-IV K1 type beta-lactamase enzymeMore data for this Ligand-Target Pair
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TargetBeta-lactamase(Enterobacter cloacae)TBA
LigandPNGBDBM50212641(Brobactam)
Affinity DataIC50:  1.78E+3nMAssay Description:Inhibitory activity against Enterobacter cloacae HC8 Class-I beta-lactamase enzyme type P99More data for this Ligand-Target Pair
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TargetBeta-lactamase(Citrobacter freundii)TBA
LigandPNGBDBM50212641(Brobactam)
Affinity DataIC50:  1.78E+3nMAssay Description:Inhibitory activity against Citrobacter freundii 87470 Class-I beta-lactamase enzymeMore data for this Ligand-Target Pair
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