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Found 2 Enz. Inhib. hit(s) with Target = 'C-C chemokine receptor type 5' and Ligand = 'BDBM50441708'
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM50441708(CHEMBL2435848)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of CCR5 (unknown origin) expressed in human HeLa cells assessed as inhibition of interaction of CHO cells expressing HIV-1 JRFLenv and HIV...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 5(Homo sapiens (Human))
Sanofi

Curated by ChEMBL
LigandPNGBDBM50441708(CHEMBL2435848)
Affinity DataIC50:  4.20nMAssay Description:Antagonist activity at CCR5 (unknown origin) expressed in HEK293F cell membranes assessed as inhibition of RANTES-induced calcium flux preincubated f...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed