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Found 3 Enz. Inhib. hit(s) with Target = 'CREB-binding protein' and Ligand = 'BDBM188516'
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

LigandPNGBDBM188516(BDOIA383)
Affinity DataIC50:  120nMAssay Description:The assay used His-tagged CBP protein, biotinylated histone H4, and detection reagents europium-labeled streptavidin and anti-6His antibody labeled w...More data for this Ligand-Target Pair
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

LigandPNGBDBM188516(BDOIA383)
Affinity DataIC50:  120nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

LigandPNGBDBM188516(BDOIA383)
Affinity DataKd:  120nMAssay Description:Experiments were performed using recombinant CBP and BRD4 bromodomainsusing the procedure reported recently (Hett et al., 2015).More data for this Ligand-Target Pair