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Found 3 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50381880'
TargetCannabinoid receptor 1(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50381880(CHEMBL2022698)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]CP55940 from recombinant human CB1 receptor expressed in human HEK293 cell membrane after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50381880(CHEMBL2022698)
Affinity DataKi:  43nMAssay Description:Displacement of [3H]CP55,940 from human recombinant CB1 receptor expressed in HEK293 cell membranes after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
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Curated by ChEMBL
LigandPNGBDBM50381880(CHEMBL2022698)
Affinity DataEC50:  1.59E+3nMAssay Description:Agonist activity at CB1 receptor in rat cerebellar membranes by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed