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Found 6 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50301311'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301311((+/-)3,3,3-trifluoro-2-methyl-N-(8-morpholino-5,6,...)
Affinity DataKi:  2.30nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301311((+/-)3,3,3-trifluoro-2-methyl-N-(8-morpholino-5,6,...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301311((+/-)3,3,3-trifluoro-2-methyl-N-(8-morpholino-5,6,...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]-CP-55940 from human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301311((+/-)3,3,3-trifluoro-2-methyl-N-(8-morpholino-5,6,...)
Affinity DataEC50:  3.60nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301311((+/-)3,3,3-trifluoro-2-methyl-N-(8-morpholino-5,6,...)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50301311((+/-)3,3,3-trifluoro-2-methyl-N-(8-morpholino-5,6,...)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells by [35S]GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed