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Found 2 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 2' and Ligand = 'BDBM50302299'
TargetCannabinoid receptor 2(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302299(2,2-dimethyl-N-(5-methyl-4-(morpholinomethyl)pyrid...)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]CP55960 from human cloned CB2 receptor after 60 mins by scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Adolor

Curated by ChEMBL
LigandPNGBDBM50302299(2,2-dimethyl-N-(5-methyl-4-(morpholinomethyl)pyrid...)
Affinity DataEC50:  4.10nMAssay Description:Agonist activity at CB2 receptor in rat cerebellar membrane assessed as WIN 55212-2-stimulated [35S]GTPgammaS binding after 6 hrs by scintillation sp...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed