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Found 1 Enz. Inhib. hit(s) with Target = 'Class D beta-lactamase' and Ligand = 'BDBM50053173'
TargetClass D beta-lactamase(Brachyspira pilosicoli)
Institut Pasteur

Curated by ChEMBL
LigandPNGBDBM50053173((2S,3S,5R)-3-Methyl-4,4,7-trioxo-3-[1,2,3]triazol-...)
Affinity DataIC50:  160nMAssay Description:Inhibition of Brachyspira pilosicoli beta-lactamase OXA-63 expressed in Escherichia coli BL21 (DE3) assessed as reduction in nitrocefin hydrolysis by...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed