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Found 3 Enz. Inhib. hit(s) with Target = 'Cyclin-A2/Cyclin-dependent kinase 2' and Ligand = 'BDBM7132'
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia Italia

LigandPNGBDBM7132(1-N-(5-cyclopropyl-1H-pyrazol-3-yl)benzene-1,4-dic...)
Affinity DataIC50:  68nMpH: 7.4 T: 2°CAssay Description:The biochemical activity of compounds was determined by incubation with specific enzymes and substrates in the presence ATP/[gamma-33P] ATP. After in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia Italia

LigandPNGBDBM7132(1-N-(5-cyclopropyl-1H-pyrazol-3-yl)benzene-1,4-dic...)
Affinity DataKd:  388nMpH: 7.5 T: 2°CAssay Description:ITCMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-A2/Cyclin-dependent kinase 2(Homo sapiens (Human))
Pharmacia Italia

LigandPNGBDBM7132(1-N-(5-cyclopropyl-1H-pyrazol-3-yl)benzene-1,4-dic...)
Affinity DataKd:  362nMpH: 7.5 T: 2°CAssay Description:OctetRedMore data for this Ligand-Target Pair
In DepthDetails PubMed