Found 3 Enz. Inhib. hit(s) with Target = 'Cyclin-dependent kinase 12' and Ligand = 'BDBM50584000' 
Affinity DataIC50: 469nMAssay Description:Inhibition of human CDK12 (696 to 1082 residues) /cyclinK (1 to 300 residues) using ac-YSPTSPpSYSPTSFpS-YSPTSPpSY-[PEG2]-RR-amid peptide as substrate...More data for this Ligand-Target Pair
3D Structure (crystal)Affinity DataKd: 98nMAssay Description:Binding affinity to partial length human wild-type CDK12 expressed in mammalian expression system assessed as dissociation constant by DiscoverX KINO...More data for this Ligand-Target Pair
Affinity DataKd: 98nMAssay Description:Binding affinity to CDK12 (unknown origin) assessed as dissociation constantMore data for this Ligand-Target Pair
