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Found 2 Enz. Inhib. hit(s) with Target = 'Cytochrome P450 3A4' and Ligand = 'BDBM151186'
TargetCytochrome P450 3A4(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM151186(US8987313, 8)
Affinity DataIC50:  170nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetCytochrome P450 3A4(Homo sapiens (Human))
Gilead Sciences

US Patent
LigandPNGBDBM151186(US8987313, 8)
Affinity DataIC50:  240nMT: 2°CAssay Description:The potencies of the compounds as inhibitors of human hepatic cytochromes P450 of the CYP3A subfamily (particularly CYP3A4) were assessed using well-...More data for this Ligand-Target Pair
In DepthDetails US Patent