Affinity DataKi: <6nMAssay Description:The binding affinity was evaluated on Dopamine receptor D2 expressed in rat striatum by using [3H]spiperone as radioligandMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Affinity DataKi: 84nMAssay Description:Binding affinity against Dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Affinity DataKi: 86nMAssay Description:Binding affinity against [3H]U-86,170-labeled dopamine receptor D2 in cloned CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 86nMAssay Description:Tested in vitro for the inhibition of [3H]-raclopride binding to Dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
Affinity DataKi: 86nMAssay Description:Displacement of [3H]-U-86,170 from Dopamine receptor D2More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Affinity DataKi: 86nMAssay Description:Binding affinity against [3H]-U-86,170-labeled dopamine receptor D2 in cloned CHO cellsMore data for this Ligand-Target Pair
Affinity DataKi: 550nMAssay Description:Displacement of [3H]YM-09151-2 from rat striatum D2 receptorMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Affinity DataKi: >1.00E+3nMAssay Description:D2 Dopamine Receptor:Radioligand binding was performed using membranes from CHO-K1 cells stably transfected with the human D2 receptor. All assays we...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against [3H]-raclopride-labeled dopamine receptor D2 in rat striatum.More data for this Ligand-Target Pair
Affinity DataKi: <1.00E+3nMAssay Description:Displacement of [3H]spiperone from rat brain Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity for [3H]raclopride-labeled dopamine receptor D2 in rat striatumMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Affinity DataKi: 1.13E+3nMAssay Description:Binding affinity against Dopamine receptor D2 from CHO-K1 cells, using [3H]-U-86,170 as the radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 1.36E+3nMAssay Description:Displacement of [3H]-spiperone from dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 1.36E+3nMAssay Description:Displacement of the radioligand [3H]-spiperone from D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.36E+3nMAssay Description:Binding affinity against D2 receptor in homogenated rat brain tissue, using by [3H]spiperone as radioligandMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Affinity DataKi: 2.38E+3nMAssay Description:Inhibition of [3H]raclopride binding to Dopamine receptor D2 of bovine striatumMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Affinity DataKi: 3.24E+3nMAssay Description:Inhibitory activity against [125I]- NCQ298 binding to dopamine receptor D2 in Sf 9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 3.50E+3nMAssay Description:Binding affinity of compound against Dopamine receptor D2 binding site using radioligand [3H]spiperoneMore data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Binding affinity to rat Dopamine receptor D2 expressed in CHO cells was determined using [125 I ] iodosulpride as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Binding affinity towards rat Dopamine receptor D2 was evaluated using [3H]- spiroperidol as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Binding affinity against D2 receptor in calf caudate nucleusMore data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Compound was evaluated for the binding affinity towards Dopamine receptor D2 using [3H]-raclopride radioligand.More data for this Ligand-Target Pair
TargetD(2) dopamine receptor(Homo sapiens (Human))
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Cooperation Pharmaceutique Fran�Aise
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibitory concentration of the compound against binding of Dopamine receptor D2 by displacement of [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataIC50: 5.76E+3nMAssay Description:In vitro binding activity against Dopamine receptor D2 from homogenized rat brain, using [3H]spiperone as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 5.80E+3nMAssay Description:The compound was tested in vitro for inhibitory activity against dopamine receptor in rats using [3H]-spiperone as radioligandMore data for this Ligand-Target Pair