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Found 2 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM50002158'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002158(5-Fluoro-3-[4-(4-phenyl-3,6-dihydro-2H-pyridin-1-y...)
Affinity DataKi:  1.60nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes [3H]ADTN, a dopamine agonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
E. Merck Darmstadt

Curated by ChEMBL
LigandPNGBDBM50002158(5-Fluoro-3-[4-(4-phenyl-3,6-dihydro-2H-pyridin-1-y...)
Affinity DataIC50:  10nMAssay Description:Evaluated for its ability to displace tritiated receptor ligand in rat striatal membranes 3[H]spiperone, a dopamine antagonistMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed