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Found 2 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM50002245'
TargetD(2) dopamine receptor(BOVINE)
New York University

Curated by ChEMBL
LigandPNGBDBM50002245(4-[2-(1-Cyclopropylmethyl-piperidin-4-yl)-acetyl]-...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity against Dopamine receptor D2 in bovine striatal homogenate using 200 pM [3H]- spiperone and 250 nM unlabeled ketanserinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Mus musculus (Mouse))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50002245(4-[2-(1-Cyclopropylmethyl-piperidin-4-yl)-acetyl]-...)
Affinity DataIC50: >1.00E+4nMAssay Description:In vitro binding affinity towards dopamine receptor D2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed