Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'D(2) dopamine receptor' and Ligand = 'BDBM50007573'
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007573(4-(1-Propyl-1,2,5,6-tetrahydro-pyridin-3-yl)-thiaz...)
Affinity DataIC50:  574nMAssay Description:Binding affinity towards dopamine receptor D2 in rat striatal membrane using [3H]spiperoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007573(4-(1-Propyl-1,2,5,6-tetrahydro-pyridin-3-yl)-thiaz...)
Affinity DataIC50:  596nMAssay Description:Inhibition of [3H]haloperidol binding for Dopamine receptor D2 in rat striatal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Rattus norvegicus (rat))
Warner-Lambert

Curated by ChEMBL
LigandPNGBDBM50007573(4-(1-Propyl-1,2,5,6-tetrahydro-pyridin-3-yl)-thiaz...)
Affinity DataIC50:  958nMAssay Description:Inhibition of [3H]haloperidol binding for Dopamine receptor D2 in rat striatal membranes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed