Affinity DataKi: 4.10nMAssay Description:Binding affinityagainst Dopamine receptor D2 in CHO-K1 cells using radioligand [3H]-NPA binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Binding affinity at Dopamine receptor D2 in rat striatal membrane by [3H]-spiperone displacement.More data for this Ligand-Target Pair
Affinity DataKi: 32.4nMAssay Description:Binding affinity towards dopamine receptor D2 of rat striatal membrane was determinedMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:In vivo Dopamine receptor D2 mitogenesis measured as [3H]-thymidine incorporation in CHO p-5 cells expressing human D2 receptorsMore data for this Ligand-Target Pair