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Found 3 Enz. Inhib. hit(s) with Target = 'D(3) dopamine receptor' and Ligand = 'BDBM50139866'
TargetD(3) dopamine receptor(Rattus norvegicus (Rat))
Aptuit

Curated by ChEMBL
LigandPNGBDBM50139866(CHEMBL3764191 | US10577361, E28)
Affinity DataKi:  100nMAssay Description:Displacement of [125I]-7-OH-PIPAT from rat brain dopamine D3 receptor after 45 mins by microplate scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(3) dopamine receptor(Homo sapiens (Human))
Indivior

US Patent
LigandPNGBDBM50139866(CHEMBL3764191 | US10577361, E28)
Affinity DataKi:  112nMAssay Description:[3H]-Spiperone Binding Assay at hD3 and hD4 recombinant receptors CHO cells transiently transfected with human dopamine type 3 or 4 receptors (CHO-hD...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetD(3) dopamine receptor(Homo sapiens (Human))
Indivior

US Patent
LigandPNGBDBM50139866(CHEMBL3764191 | US10577361, E28)
Affinity DataKi: <1.00E+4nMAssay Description:Agonist activity at human dopamine D3 receptor expressed in CHO cells after 90 mins by [35S]-GTPgamma S assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed