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Found 4 Enz. Inhib. hit(s) with Target = 'DNA-dependent protein kinase catalytic subunit' and Ligand = 'BDBM50132361'
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132361(2-(4-Methoxy-phenyl)-6-morpholin-4-yl-pyran-4-one ...)
Affinity DataIC50:  220nMAssay Description:In vitro inhibition of DNA-dependent protein kinase(DNA-PK) from HeLa (human carcinoma) cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132361(2-(4-Methoxy-phenyl)-6-morpholin-4-yl-pyran-4-one ...)
Affinity DataIC50:  220nMAssay Description:Inhibition of DNA-PK (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132361(2-(4-Methoxy-phenyl)-6-morpholin-4-yl-pyran-4-one ...)
Affinity DataIC50:  220nMAssay Description:Inhibition of DNA-PK in HeLa cell nuclear extractsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA-dependent protein kinase catalytic subunit(Homo sapiens (Human))
University Of Newcastle

Curated by ChEMBL
LigandPNGBDBM50132361(2-(4-Methoxy-phenyl)-6-morpholin-4-yl-pyran-4-one ...)
Affinity DataIC50:  220nMAssay Description:Inhibition of DNA-PKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed