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Found 3 Enz. Inhib. hit(s) with Target = 'Dipeptidyl peptidase 4' and Ligand = 'BDBM11159'
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM11159((1R)-1-(3,4-difluorobenzyl)-3-oxo-3-[3-(trifluorom...)
Affinity DataIC50:  128nMpH: 7.5 T: 2°CAssay Description:The enzyme activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 360 nm and m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM11159((1R)-1-(3,4-difluorobenzyl)-3-oxo-3-[3-(trifluorom...)
Affinity DataIC50:  128nMAssay Description:Inhibition of DPP4 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM11159((1R)-1-(3,4-difluorobenzyl)-3-oxo-3-[3-(trifluorom...)
Affinity DataIC50:  128nMAssay Description:Inhibition of DPP4 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed