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Found 3 Enz. Inhib. hit(s) with Target = 'Dual specificity tyrosine-phosphorylation-regulated kinase 1A' and Ligand = 'BDBM80396'
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM80396((1E)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylide...)
Affinity DataIC50:  12nMAssay Description:Inhibition of Dyrk1A kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM80396((1E)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylide...)
Affinity DataIC50:  930nMAssay Description:Inhibition of DYRK1A (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
National Human Genome Research Institute

Curated by ChEMBL
LigandPNGBDBM80396((1E)-1-(3-ethyl-5-methoxy-1,3-benzothiazol-2-ylide...)
Affinity DataKd:  12nMAssay Description:Binding affinity to Dyrk1A assessed as dissociation constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed