Found 1 Enz. Inhib. hit(s) with Target = 'E3 ubiquitin-protein ligase Mdm2' and Ligand = 'BDBM50165718'
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 334nMAssay Description:Binding affinity to human MDM2 assessed as inhibition of interaction with p53 by fluorescence polarization assayMore data for this Ligand-Target Pair