Affinity DataIC50: 1.56E+4nMAssay Description:Displacement of [125I]ET1 from human ETB receptor expressed in membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1.56E+4nMAssay Description:Antagonist activity at ETB receptor (unknown origin) expressed in HEK293T cells measured after 30 mins by CCF4-AM dye based GeneBlazer FRET assayMore data for this Ligand-Target Pair