Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Estrogen receptor beta' and Ligand = 'BDBM19966'
TargetEstrogen receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM19966(6-(4-methanesulfonylphenyl)-5-{4-[2-(piperidin-1-y...)
Affinity DataKi:  1.32nMAssay Description:Displacement of [3H]estradiol from human recombinant ERbetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM19966(6-(4-methanesulfonylphenyl)-5-{4-[2-(piperidin-1-y...)
Affinity DataKi:  1.36nM ΔG°:  -50.1kJ/mole EC50:  10.7nMpH: 7.5 T: 2°CAssay Description:The binding affinities were determined by a competitive radiometric binding assay using [3H]estradiol as tracer. The Kd for 3H-estradiol was determin...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed