Affinity DataIC50: 9.10nMAssay Description:Inhibition of human FAK using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of FAK (unknown origin) by Lanthascreen assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of human FAK using poly[Glu:Tyr] (4:1) as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of FAK (unknown origin) after 40 mins by scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of human FAK/PTK2 using poly[Glu:Tyr] (4:1) as substrate in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
Affinity DataIC50: 55nMAssay Description:Inhibition of human FAK by kinase inhibition assayMore data for this Ligand-Target Pair
Affinity DataIC50: 62nMAssay Description:Inhibition of recombinant human FAK expressed in Sf9 insect cells using Ulight-TK peptide as substrate after 60 mins by LANCE methodMore data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of FAK (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of FAK (unknown origin) assembly after 20 mins by turbidimetric methodMore data for this Ligand-Target Pair
Affinity DataIC50: 3.12E+3nMAssay Description:Inhibition of full-length Homo sapiens (human) recombinant FAK assessed as remaining ATP content after 4 hr by Kinase-Glo luminescence analysisMore data for this Ligand-Target Pair
Affinity DataKd: 64nMAssay Description:Binding constant for FAK kinase domainMore data for this Ligand-Target Pair
Affinity DataKd: 68nMAssay Description:Average Binding Constant for PTK2; NA=Not Active at 10 uMMore data for this Ligand-Target Pair
Affinity DataEC50: 2.35E+4nMAssay Description:Inhibition of human recombinant full-length FAK assessed as remaining ATP after 4 hrs by Kinase-Glo-luminescence assayMore data for this Ligand-Target Pair
Affinity DataKd: 64nMAssay Description:Binding constant for PTK2 kinase domainMore data for this Ligand-Target Pair