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Found 3 Enz. Inhib. hit(s) with Target = 'GABA-A receptor; alpha-5/beta-3/gamma-2' and Ligand = 'BDBM50034820'
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
University Of Wisconsin-Milwaukee

Curated by ChEMBL
LigandPNGBDBM50034820(8-Chloro-3-methoxymethyl-5-methyl-4,5-dihydro-2,5,...)
Affinity DataKi:  39nMAssay Description:Binding affinity for Gamma-aminobutyric-acid A receptor alpha5-beta3-gamma2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
University Of Wisconsin-Milwaukee

Curated by ChEMBL
LigandPNGBDBM50034820(8-Chloro-3-methoxymethyl-5-methyl-4,5-dihydro-2,5,...)
Affinity DataKi:  39nMAssay Description:Binding affinity for human recombinant gamma-aminobutyric-acid (GABA) A receptor alpha-5-beta-3-gamma-2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGABA-A receptor; alpha-5/beta-3/gamma-2(Homo sapiens (Human))
University Of Wisconsin-Milwaukee

Curated by ChEMBL
LigandPNGBDBM50034820(8-Chloro-3-methoxymethyl-5-methyl-4,5-dihydro-2,5,...)
Affinity DataKi: >300nMAssay Description:Binding affinity to human recombinant GABA alpha5beta3gamma2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed