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Found 5 Enz. Inhib. hit(s) with Target = 'Gag-Pol polyprotein [489-587]' and Ligand = 'BDBM50014151'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50014151(((1S,2R,3R,4S)-1-Benzyl-4-tert-butoxycarbonylamino...)
Affinity DataKi:  40nMAssay Description:Binding affinity to HIV-1 proteaseChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50014151(((1S,2R,3R,4S)-1-Benzyl-4-tert-butoxycarbonylamino...)
Affinity DataIC50:  40nMAssay Description:Inhibitory activity against recombinant HIV-1 ProteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50014151(((1S,2R,3R,4S)-1-Benzyl-4-tert-butoxycarbonylamino...)
Affinity DataIC50:  280nMAssay Description:Inhibition of HIV-1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50014151(((1S,2R,3R,4S)-1-Benzyl-4-tert-butoxycarbonylamino...)
Affinity DataIC50:  1.38E+3nMAssay Description:Inhibition of HIV-1 protease was determined in vitroChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50014151(((1S,2R,3R,4S)-1-Benzyl-4-tert-butoxycarbonylamino...)
Affinity DataIC50:  1.38E+3nMAssay Description:Inhibitory activity against HIV-1 protease.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed