Found 5 Enz. Inhib. hit(s) with Target = 'Gamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2' and Ligand = 'BDBM26266' TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Rattus norvegicus (Rat))
University Of Firenze
Curated by ChEMBL
University Of Firenze
Curated by ChEMBL
Affinity DataKi: 156nMAssay Description:Binding affinity for recombinant rat GABA-A receptor alpha2-beta2-gamma2 subunits expressed in HEK293 cellsMore data for this Ligand-Target Pair
3D Structure (crystal)TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Rattus norvegicus (Rat))
University Of Firenze
Curated by ChEMBL
University Of Firenze
Curated by ChEMBL
Affinity DataKi: 765nMAssay Description:Displacement of [3H]flumazenil from rat GABA-Aalpha2 receptor plus beta-2-gamma-2 in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Rattus norvegicus (Rat))
University Of Firenze
Curated by ChEMBL
University Of Firenze
Curated by ChEMBL
Affinity DataKi: 765nMAssay Description:Displacement of [3H]-flumazenil from rat GABA-A Gamma-aminobutyric acid A receptor alpha2-beta2-gamma2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Rattus norvegicus (Rat))
University Of Firenze
Curated by ChEMBL
University Of Firenze
Curated by ChEMBL
Affinity DataKi: 765nMAssay Description:Displacement of [3H]flumazenil from rat GABAA alpha2beta2gamma2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetGamma-aminobutyric acid receptor subunit alpha-2/beta-2/gamma-2(Homo sapiens (Human))
Universit£
Curated by ChEMBL
Universit£
Curated by ChEMBL
Affinity DataEC50: 1.80E+9nMAssay Description:Potentiation of GABA-evoked Cl- currents in Xenopus oocytes expressing human alpha-2-beta-2-gamma-2 subunitsMore data for this Ligand-Target Pair
