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Found 1 Enz. Inhib. hit(s) with Target = 'Geranylgeranyl transferase type-1 subunit beta/Protein farnesyltransferase/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50134309'
LigandPNGBDBM50134309(2-Methyl-2,3,10,10a-tetrahydro-pyrazino[1,2-a]indo...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of [3H]-GGPP incorporation into recombinant human Ha-Ras-CVLL by Geranylgeranyl transferase type IMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed