Affinity DataKi: 7.10nMAssay Description:Binding affinity for glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 95nMAssay Description:Binding affinity for glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 95nMAssay Description:Binding affinity for glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 1.30nMAssay Description:Transcriptional repression of IL-1 stimulated IL-6 expression in native cells compared to dexamethasoneMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Repression activity of GR ligand with interleukin-6 receptor in native cell assay using dexamethasone was determined as maximal potencyMore data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Transcriptional repression activity in HEP G2 cells expressing glucocorticoid receptor compared to dexamethasoneMore data for this Ligand-Target Pair
Affinity DataIC50: 107nMAssay Description:Transcriptional activation in CV-1 cells expressing glucocorticoid receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 139nMAssay Description:Glucocorticoid-induced aromatase activity in human skin fibroblastsMore data for this Ligand-Target Pair