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Found 4 Enz. Inhib. hit(s) with Target = 'Glucocorticoid receptor' and Ligand = 'BDBM50144471'
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144471(CHEMBL68083 | N-{3-[Benzyl-(2,4-difluoro-benzyl)-a...)
Affinity DataIC50:  15nMAssay Description:Binding affinity against human Glucocorticoid receptor (GR) using [3H]-dexamethasone as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144471(CHEMBL68083 | N-{3-[Benzyl-(2,4-difluoro-benzyl)-a...)
Affinity DataIC50:  15nMAssay Description:Inhibition of [3H]dexamethasone binding to human glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144471(CHEMBL68083 | N-{3-[Benzyl-(2,4-difluoro-benzyl)-a...)
Affinity DataIC50:  100nMAssay Description:Inhibition of glucocorticoid receptor Dexamethasone response in reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50144471(CHEMBL68083 | N-{3-[Benzyl-(2,4-difluoro-benzyl)-a...)
Affinity DataIC50:  100nMAssay Description:Functional activity towards human Glucocorticoid receptor in genetically engineered cell line containing glucocorticoid response element and reporter...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed