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Found 4 Enz. Inhib. hit(s) with Target = 'Glucocorticoid receptor' and Ligand = 'BDBM50259979'
TargetGlucocorticoid receptor(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259979(CHEMBL4090392)
Affinity DataIC50:  6.30nMAssay Description:Transrepression activity at glucocorticoid receptor in human THP1 cells assessed as receptor-mediated anti-inflammatory activity by measuring inhibit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259979(CHEMBL4090392)
Affinity DataIC50:  6.30nMAssay Description:Transactivation activity at glucocorticoid receptor in human HeLa cells assessed as induction of MMTV promoter activity by luciferase reporter gene a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259979(CHEMBL4090392)
Affinity DataIC50:  25nMAssay Description:Transactivation activity at glucocorticoid receptor in human HeLa cells assessed as induction of MMTV promoter activity by luciferase reporter gene a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Bayer Pharma

Curated by ChEMBL
LigandPNGBDBM50259979(CHEMBL4090392)
Affinity DataIC50:  126nMAssay Description:Transactivation activity at glucocorticoid receptor in human HeLa cells assessed as induction of MMTV promoter activity by luciferase reporter gene a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed