Found 2 Enz. Inhib. hit(s) with Target = 'Glucose-dependent insulinotropic receptor' and Ligand = 'BDBM50240388'
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: 1.80nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Jiangxi University of Traditional Chinese Medicine
Curated by ChEMBL
Jiangxi University of Traditional Chinese Medicine
Curated by ChEMBL
Affinity DataEC50: 5.30nMAssay Description:Agonist activity at human GPR119 expressed in HEK293 cells assessed as increase in cAMP stimulation measured after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair