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Found 3 Enz. Inhib. hit(s) with Target = 'Glucose-dependent insulinotropic receptor' and Ligand = 'BDBM50315136'
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50315136(CHEMBL1092240 | N-(4-(1H-1,2,4-triazol-1-yl)phenyl...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human GPR119 receptor by cAMP mobilization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50315136(CHEMBL1092240 | N-(4-(1H-1,2,4-triazol-1-yl)phenyl...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human GPR119 receptor expressed in CHO-K1 cells co-expressing 6CRE-luciferase gene after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucose-dependent insulinotropic receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50315136(CHEMBL1092240 | N-(4-(1H-1,2,4-triazol-1-yl)phenyl...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at GPR119 receptor by cell based cAMP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed