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Found 1 Enz. Inhib. hit(s) with Target = 'Glutamate receptor ionotropic, kainate 5' and Ligand = 'BDBM50207594'
TargetGlutamate receptor ionotropic, kainate 5(Rattus norvegicus)
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Curated by ChEMBL
LigandPNGBDBM50207594(2,3-Dihydroxy-6-nitro-benzo[f]quinoxaline-7-sulfon...)
Affinity DataKd:  1.78E+3nMAssay Description:Antagonist activity against GLUK5-containing kainate receptor by inhibition of kainate-induced depolarization of neonatal rat dorsal root fibersMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed