Found 1 Enz. Inhib. hit(s) with Target = 'HLA class II histocompatibility antigen gamma chain/Proto-oncogene tyrosine-protein kinase ROS' and Ligand = 'BDBM50018830'
TargetHLA class II histocompatibility antigen gamma chain/Proto-oncogene tyrosine-protein kinase ROS(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: 0.230nMAssay Description:Inhibition of CD74-ROS1 (unknown origin) expressed in mouse BaF3 cells assessed as reduction in cell viabilityMore data for this Ligand-Target Pair