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Found 4 Enz. Inhib. hit(s) with Target = 'Heparanase' and Ligand = 'BDBM50165652'
TargetHeparanase(Homo sapiens (Human))
Sharif University Of Technology

Curated by ChEMBL
LigandPNGBDBM50165652((2-{4-[3-((E)-4-Bromo-phenyl)-acryloylamino]-3-flu...)
Affinity DataIC50:  398nMAssay Description:Inhibition of heparanaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Sharif University Of Technology

Curated by ChEMBL
LigandPNGBDBM50165652((2-{4-[3-((E)-4-Bromo-phenyl)-acryloylamino]-3-flu...)
Affinity DataIC50:  400nMAssay Description:Inhibition of human heparanase assessed as reduction in basic fibroblast growth factor binding incubated for 2 hrs by microplate reader assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHeparanase(Homo sapiens (Human))
Sharif University Of Technology

Curated by ChEMBL
LigandPNGBDBM50165652((2-{4-[3-((E)-4-Bromo-phenyl)-acryloylamino]-3-flu...)
Affinity DataIC50:  400nMAssay Description:In vitro inhibitory concentration against human HeparanaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHeparanase(Homo sapiens (Human))
Sharif University Of Technology

Curated by ChEMBL
LigandPNGBDBM50165652((2-{4-[3-((E)-4-Bromo-phenyl)-acryloylamino]-3-flu...)
Affinity DataIC50:  7.68E+3nMAssay Description:Recombinant human active heparanase derived from Chinese hamster ovary cells was from R&D Systems. Bovine serum albumin-coated 96 well microplates (9...More data for this Ligand-Target Pair
In DepthDetails US Patent