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Found 3 Enz. Inhib. hit(s) with Target = 'Histamine H3 receptor' and Ligand = 'BDBM50212733'
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50212733(CHEMBL425994 | N-(2-((dimethylamino)methyl)-4-(3-(...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity to human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50212733(CHEMBL425994 | N-(2-((dimethylamino)methyl)-4-(3-(...)
Affinity DataKi:  9.80nMAssay Description:Binding affinity to rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50212733(CHEMBL425994 | N-(2-((dimethylamino)methyl)-4-(3-(...)
Affinity DataEC50:  0.200nMAssay Description:Inverse agonist activity at human histamine H3 receptor by GTP gammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed