Affinity DataKi: 0.126nMAssay Description:Displacement of [3H]N-alpha-Methylhistamine from human recombinant H3 receptor expressed in HEK293 cells by competitive binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.316nMAssay Description:Binding affinity to human histamine H3 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 2.51nMAssay Description:Inverse agonist activity at human histamine H3 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair