Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Histamine H4 receptor' and Ligand = 'BDBM26395'
TargetHistamine H4 receptor(Rattus norvegicus (rat))
Abbott Laboratories

LigandPNGBDBM26395(2,4-diamino-5,6-disubstituted pyrimidine, 9 | 6-(p...)
Affinity DataKi:  7.60nM ΔG°:  -46.3kJ/molepH: 7.4 T: 2°CAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM26395(2,4-diamino-5,6-disubstituted pyrimidine, 9 | 6-(p...)
Affinity DataKi:  71nM ΔG°:  -40.8kJ/molepH: 7.4 T: 2°CAssay Description:Competition radioligand binding assays were performed with increasing concentrations of test compound in the presence of [3H]ligand. All binding reac...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Abbott Laboratories

LigandPNGBDBM26395(2,4-diamino-5,6-disubstituted pyrimidine, 9 | 6-(p...)
Affinity DataKi:  79.4nMAssay Description:Binding affinity to H4R receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed