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Found 2 Enz. Inhib. hit(s) with Target = 'Histone acetyltransferase GCN5' and Ligand = 'BDBM50076253'
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50076253(CHEMBL3416314)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of Vps75-stimulated recombinant Saccharomyces cerevisiae histone acetyltransferase Rtt109 using Asf1-dH3-H4 as substrate assessed as coenz...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Mayo Clinic

Curated by ChEMBL
LigandPNGBDBM50076253(CHEMBL3416314)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of Vps75-stimulated recombinant Saccharomyces cerevisiae histone acetyltransferase Rtt109 using Asf1-dH3-H4 as substrate assessed as coenz...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed