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Found 1 Enz. Inhib. hit(s) with Target = 'Histone deacetylase 8' and Ligand = 'BDBM152730'
TargetHistone deacetylase 8(Homo sapiens (Human))
University of Pennsylvania

LigandPNGBDBM152730(7-Amino-N-hydroxypentanamide (6))
Affinity DataIC50:  5.30E+3nMpH: 8.2Assay Description:Activity assays were conducted at 25 °C and contained 500 nM HDAC8 enzyme, 150 μM Ac-Arg-His-Lys(Ac)-Lys(Ac)-aminomethylcoumarin substrate (BML-...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed