Found 1 Enz. Inhib. hit(s) with Target = 'Histone-lysine N-methyltransferase 2A' and Ligand = 'BDBM50601692'
TargetHistone-lysine N-methyltransferase 2A(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 190nMAssay Description:Inhibition of MLL1 (unknown origin) histone methyltransferase activityMore data for this Ligand-Target Pair